阿替美唑盐酸盐酸盐是一种有效的肾上腺素受体阻断药，其选择性和竞争性的抑制肾上腺素受体。在作为兽药方面，阿替美唑盐酸盐酸盐主要用于牲畜，如狗，在手术后，使其迅速的从使用麻醉药物肾上腺素受体激动剂美托咪叮所产生的镇静及其他一些作用中恢复。对狗肌肉注射该药后，分钟即可起效，分钟左右达到血糖浓度而其在血液中的半衰期小于小时，随后通过在肝脏内进行生物转化，经尿液排出。由此可见阿替美唑盐酸盐酸盐是一种有效快捷安全的药物。Atamezole hydrochloride is an effective adrenergic receptor blocker that selectively and competitively inhibits adrenergic receptors. As a veterinary drug, atamezole hydrochloride is primarily used in livestock, such as dogs, after surgery to quickly recover from the sedative effects and other actions of the adrenergic receptor agonist medetomidine. After intramuscular injection in dogs, it takes effect within minutes, reaches its blood concentration in about 10 minutes, and has a half-life of less than one hour in the bloodstream. It is then biotransformed in the liver and excreted through urine. This demonstrates that atamezole hydrochloride is an effective, fast-acting, and safe medication.
