5-Bromo-2-chloro-pyrimidine;5-Hydroxy-pyridine-2-carboxylic acid methyl ester;(2R,5S)-1-Boc-2,5-dimethyl-piperazine;6-Bromo-1H-indazole;cis-4-Amino-cyclohexanol hydrochloride;4-Methyl-6-trifluoromethyl-pyridin-2-ol;5-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-oxazole;(1R,3R,5R)-2-Boc-2-aza-bicyclo[3.1.0]hexane-3-dicarboxylic acid;5-Bromo-2-chloro-pyrimidine;5-Hydroxy-pyridine-2-carboxylic acid methyl ester;(2R,5S)-1-Boc-2,5-dimethyl-piperazine;6-Bromo-1H-indazole;cis-4-Amino-cyclohexanol hydrochloride;4-Methyl-6-trifluoromethyl-pyridin-2-ol;5-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-oxazole;(1R,3R,5R)-2-Boc-2-aza-bicyclo[3.1.0]hexane-3-dicarboxylic acid;2,6-Dichloro-benzamidine hydrochloride;4-Methoxy-2-methyl-piperidine hydrochloride;Octahydro-[1,6]naphthyridine-1-carboxylic acid tert-butyl ester hydrochloride;(1-Methyl-3-oxo-cyclopentyl)-carbamic acid tert-butyl ester;Methyl-(tetrahydro-pyran-2-ylmethyl)-amine;2-Methyl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-oxazole;(R)-Tetrahydro-pyran-3-carboxylic acid;1,1-Dioxo-hexahydro-1l6-thiopyran-3-ylamine;2-(Pentafluorosulfur)aniline;2,7-Dimethyl-imidazo[1,2-a]pyridine-3-carbaldehyde;5-Methyl-tetrahydro-furan-3-ol;6-Bromo-benzooxazole-2-carboxylic acid;trans-3-Amino-cyclohexyl-methanol hydrochloride;3-Bromo-2-(2,2,2-trifluoro-ethoxy)-pyridine;3-Methyl-indan-1-ylamine;5-Bromo-oxazole-2-carbaldehyde;2-Methyl-4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridine dihydrochloride;Octahydro-[1]pyrindine;N2-methyl-2-methyl-propane-1,2-diamine;5-Bromo-oxazole-2-carboxylic acid methyl ester;1,4-Dioxa-8-aza-spiro[4.6]undecane;5-Aminomethyl-1-methyl-pyrrolidin-2-one;2-(4-BROMOPHENYL)-4-(CHLOROMETHYL)-1,3-OXAZOLE;rel-(3aS,4S,7aR)-2-Boc-4-amino-octahydro-isoindole;2,6-Dichloro-benzamidine hydrochloride;4-Methoxy-2-methyl-piperidine hydrochloride;Octahydro-[1,6]naphthyridine-1-carboxylic acid tert-butyl ester hydrochloride;(S)-2-(1-Methyl-pyrrolidin-2-yl)-ethanol;1,3-Dimethyl-piperazin-2-one hydrochloride;(R)-Tetrahydro-pyran-3-carboxylic acid;trans-2-Ethyl-cyclopropylamine hydrochloride;4-Pyrrolidin-1-ylmethyl-aniline;5-Bromo-2-methyl-oxazole hydrochloride;4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-oxazole;2,2-Dimethyl-piperidine hydrochloride;N-[[4-[trifluoromethyl]-3-pyridinyl]carbonyl]-glycine;Isothiazole-4-carbaldehyde;C-(5-Cyclopropyl-1H-pyrazol-3-yl)-methylamine hydrochloride;5-Methyl-oxazole-2-carboxylic acid;3,3-Difluoro-2,2-dimethyl-propionaldehyde;1,9-Diaza-spiro[5.5]undecane-1-carboxylic acid tert-butyl ester hydrochloride;2,2,6,6-Tetramethyl-1,2,3,6-tetrahydro-4-pyridineboronic acid pinacol ester hydrochloride;(5-methyl-1,3-oxazol-4-yl)methanamine hydrochloride;4-Hydroxymethyl-oxazole-2-carboxylic acid;Imidazo[1,2-a]pyridin-3-ylmethyl-methyl-amine;4-Methyl-piperazine-1,2-dicarboxylic acid 1-tert-butyl ester;4-(2-Dimethylamino-ethyl)-aniline;2-Methyl-5,6-dihydro-4H-pyrrolo[3,4-d]thiazole hydrochloride;1-Cbz-4-(methoxy-methyl-carbamoyl)-piperidine;Isoxazol-3-yl-acetic acid;3-Trifluoromethyl-cyclopent-2-enone;1-Thiazol-4-yl-ethylamine;6-Fluoro-1H-benzoimidazole-2-carboxylic acid;1-Benzyl-piperazin-2-one;4-Ethynyl-pyrimidine;1-Methyl-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridine;5-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-2-trifluoromethyl-oxazole;2,6-Dichloro-benzamidine hydrochloride;4-Methoxy-2-methyl-piperidine hydrochloride;Octahydro-[1,6]naphthyridine-1-carboxylic acid tert-butyl ester hydrochloride;(1-Methyl-3-oxo-cyclopentyl)-carbamic acid tert-butyl ester;Methyl-(tetrahydro-pyran-2-ylmethyl)-amine;2-Methyl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-oxazole;(R)-Tetrahydro-pyran-3-carboxylic acid;1,1-Dioxo-hexahydro-1l6-thiopyran-3-ylamine;2-(Pentafluorosulfur)aniline;2,7-Dimethyl-imidazo[1,2-a]pyridine-3-carbaldehyde;5-Methyl-tetrahydro-furan-3-ol;6-Bromo-benzooxazole-2-carboxylic acid;trans-3-Amino-cyclohexyl-methanol hydrochloride;3-Bromo-2-(2,2,2-trifluoro-ethoxy)-pyridine;3-Methyl-indan-1-ylamine;5-Bromo-oxazole-2-carbaldehyde;2-Methyl-4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridine dihydrochloride;Octahydro-[1]pyrindine;N2-methyl-2-methyl-propane-1,2-diamine;5-Bromo-oxazole-2-carboxylic acid methyl ester;2-Boc-4-amino-octahydro-isoindole;1,4-Dioxa-8-aza-spiro[4.6]undecane;5-Aminomethyl-1-methyl-pyrrolidin-2-one;2-(4-BROMOPHENYL)-4-(CHLOROMETHYL)-1,3-OXAZOLE